From Flat to 3D: Replacing Phenyl Rings with Saturated Bridged Bicyclic Mimetics to Mitigate Bioactivation and Optimize ADME Properties and Oral Bioavailability in Reverse Amide Orientation
Murugaiah A. M. Subbaiah·Prakash Vachaspati·Gaurav Saini·Lavanya Billava Ramappa·Sivashankaran Raju·Joyson Nandha·Himangshu Bhowmik·Enugurthi Hari Krishna·Sushmita Janrao·V. Anil Kumar·S. Choubey·Joothipriya Subramanian·Bhuvaneshwaran Anandamoorthy·Sukanta Kumar Sahoo·Raghavendra Veerapuram·Korlepara Vamsi Krishna·Manohar Yelleswarapu·Y.K. Gupta·Muthalagu Vetrichelvan·Anuradha Gupta·Salil D. Desai·Thanga Mariappan·Arvind Mathur·Shruti Surendran