Chiral organosilicon compounds featuring a silicon-stereogenic center have attracted renewed interest in recent years. However, the enantioselective synthesis of such molecules containing both carbon and silicon stereocenters from prochiral precursors remains a significant challenge. Herein, we report a desymmetrization strategy that enables the simultaneous construction of two adjacent stereocenters at silicon and carbon. This transformation is achieved through the enantioselective copper-catal
Copper-Catalyzed Enantioselective Conjugate Borylation of Silacyclohexadienones to Construct Highly Congested Stereocenters Adjacent to C−Si Bonds
Jun-Han Ma·Li-Wen Xu·Ting Wu·Chen-Li Jin·Fei Ye·Zheng Xu·L Li·Zhi-Yuan Zhao·Martin Oestreich·Shuang-Li Liu
